Lenacapavir Naloxegol

Sunlenca Product Label

Interaction Color Code
Clinical Bottom Line
Minimal data to guide interaction: risks likely to outweigh benefits
Drug 1
Drug 2
Mechanism
Inhibition of CYP3A4 by lenacapavir
Clinical Effects

Increased risk of naloxegol adverse effects

Management

Consider using alternative agents. If coadministration is unavoidable, decrease dose of naloxegol and monitor for adverse reactions.