Etravirine Fluconazole 522

Interaction Color Code
Clinical Bottom Line
Administer standard doses
Drug 1
Drug 1 dose
200 mg BID
Drug 1 effect

Etravirine AUC increased 86%; Cmax increased 75%; Cmin increased 109%

Drug 2
Drug 2 dose
200 mg QAM
Drug 2 effect

No significant change

Clinical Effects

Increased etravirine effects

Management

Monitor for fluconazole associated toxicities

Import ID
522