Atazanavir Proguanil 853

Reyataz label

Clinical Bottom Line
Minimal data to guide interaction: weigh risks and benefits of using this combination
Drug 1
Drug 1 dose
300 mg with 100 mg ritonavir daily
Drug 1 effect

Not reported

Drug 2
Drug 2 dose
100 mg with 250 mg atovaquone x 1
Drug 2 effect

Proguanil AUC decreased 41%, Cmax no significant change

Clinical Effects

Potentially compromised antimalarial activity

Management

If coadministering monitor for anti-malarial efficacy

Import ID
853