Atazanavir Atovaquone 851

Reyataz label

Clinical Bottom Line
Minimal data to guide interaction: weigh risks and benefits of using this combination
Drug 1
Drug 1 dose
300 mg with 100 mg ritonavir daily
Drug 1 effect

Not reported

Drug 2
Drug 2 dose
250 mg with 100 mg proguanil x 1
Drug 2 effect

Atovaquone AUC decreased 46%, Cmax decreased 49%

Clinical Effects

Potential compromised antimalarial activity

Management

Dose adjustment not established. If coadministering monitor for anti-malarial efficacy.

Import ID
851