Etravirine ATV 574

Drug 1
Drug 1 effect

Etravirine AUC increased 30%; Cmax increased 30%; Cmin decreased 26%

Drug 2
Drug 2 dose
300 mg daily with 100 mg ritonavir daily
Drug 2 effect

Atazanavir AUC decreased 14%; Cmin decreased 38%

Clinical Effects

Potential for increased etravirine effects

Management

When using atazanavir 300 mg plus ritonavir 100 mg once daily use etravirine standard dose.

Import ID
574